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This is a list of steroidal estrogens or derivatives of estradiol, estrone, and estriol. Most esters of these estrogens are not included in this list; for esters, see here instead.
Estradiol derivatives
17α-Substituted estradiol derivatives
Nitrogen mustard-coupled alkylating antineoplastic estradiol derivatives
Compound
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Chemical name
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Structure
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Marketed
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Alestramustine
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Estradiol 3-(bis(2-chloroethyl)carbamate) 17β-(2β-aminopropanoate)
|
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–
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Atrimustine
|
Estradiol 3-benzoate 17β-(4-(4-(bis(2-chloroethyl)amino)phenyl)-1-oxobutoxy)acetate
|
|
–
|
Estramustine
|
Estradiol 3-(bis(2-chloroethyl)carbamate)
|
|
–
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Estramustine phosphate
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Estradiol 3-(bis(2-chloroethyl)carbamate) 17β-phosphate
|
|
✓
|
17β-Aminoestrogens
Compound
|
Chemical name
|
Structure
|
Marketed
|
Aminoestradiol
|
17β-Aminoestradiol
|
|
–
|
Butolame
|
17β-((4-Hydroxybutyl)amino)estradiol
|
|
–
|
Hexolame
|
17β-((6-Hydroxyhexyl)amino)estradiol
|
|
–
|
Pentolame
|
17β-((5-Hydroxypentyl)amino)estradiol
|
|
–
|
Prodiame
|
17β-((3-Aminopropyl)amino)estradiol
|
|
–
|
Prolame
|
17β-((3-Hydroxypropyl)amino)estradiol
|
|
–
|
Estrone derivatives
Nitrogen mustard-coupled alkylating antineoplastic estrone derivatives
Compound
|
Chemical name
|
Structure
|
Marketed
|
Estromustine
|
Estrone 3-(bis(2-chloroethyl)carbamate)
|
|
–
|
Estriol derivatives
17α-Substituted estriol derivatives
Other estrogen derivatives
Epimers
Equine estrogens
See also
Notes
? = Chemical names that are unverified.
References
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Estrogens | ERTooltip Estrogen receptor agonists |
- Steroidal: Alfatradiol
- Certain androgens/anabolic steroids (e.g., testosterone, testosterone esters, methyltestosterone, metandienone, nandrolone esters) (via estrogenic metabolites)
- Certain progestins (e.g., norethisterone, noretynodrel, etynodiol diacetate, tibolone)
- Clomestrone
- Cloxestradiol acetate
- Conjugated estriol
- Conjugated estrogens
- Epiestriol
- Epimestrol
- Esterified estrogens
- Estetrol†
- Estradiol
- Estradiol esters (e.g., estradiol acetate, estradiol benzoate, estradiol cypionate, estradiol enanthate, estradiol undecylate, estradiol valerate, polyestradiol phosphate, estradiol ester mixtures (Climacteron))
- Estramustine phosphate
- Estriol
- Estriol esters (e.g., estriol succinate, polyestriol phosphate)
- Estrogenic substances
- Estrone
- Estrone esters
- Ethinylestradiol#
- Hydroxyestrone diacetate
- Mestranol
- Methylestradiol
- Moxestrol
- Nilestriol
- Prasterone (dehydroepiandrosterone; DHEA)
- Promestriene
- Quinestradol
- Quinestrol
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Progonadotropins | |
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Antiestrogens | ERTooltip Estrogen receptor antagonists (incl. SERMsTooltip selective estrogen receptor modulators/SERDsTooltip selective estrogen receptor downregulators) | |
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Aromatase inhibitors | |
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Antigonadotropins |
- Androgens/anabolic steroids (e.g., testosterone, testosterone esters, nandrolone esters, oxandrolone, fluoxymesterone)
- D2 receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride)
- GnRH agonists (e.g., leuprorelin, goserelin)
- GnRH antagonists (e.g., cetrorelix, elagolix)
- Progestogens (e.g., chlormadinone acetate, cyproterone acetate, gestonorone caproate, hydroxyprogesterone caproate, medroxyprogesterone acetate, megestrol acetate)
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Others | |
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